In Vitro Activation of Cytochrome P450 46A1 (CYP46A1) by Efavirenz-Related Compounds.

Mast N, Verwilst P, Wilkey CJ, Guengerich FP, Pikuleva IA
J Med Chem. 2020 63 (12): 6477-6488

PMID: 31617715 · PMCID: PMC7226586 · DOI:10.1021/acs.jmedchem.9b01383

MeSH Terms (13)

Alkynes Allosteric Site Benzoxazines Catalytic Domain Cholesterol Cholesterol 24-Hydroxylase Cyclopropanes Cytochrome P-450 CYP3A Inducers Humans Hydroxylation In Vitro Techniques Pharmaceutical Preparations Protein Conformation

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