Discovery of 4-alkoxy-6-methylpicolinamide negative allosteric modulators of metabotropic glutamate receptor subtype 5.

Felts AS, Bollinger KA, Brassard CJ, Rodriguez AL, Morrison RD, Scott Daniels J, Blobaum AL, Niswender CM, Jones CK, Conn PJ, Emmitte KA, Lindsley CW
Bioorg Med Chem Lett. 2019 29 (1): 47-50

PMID: 30446311 · PMCID: PMC6295259 · DOI:10.1016/j.bmcl.2018.11.017

MeSH Terms (11)

Allosteric Regulation Animals Dose-Response Relationship, Drug Drug Discovery Humans Ligands Molecular Structure Picolinic Acids Rats Receptor, Metabotropic Glutamate 5 Structure-Activity Relationship

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