Optimization of the choline transporter (CHT) inhibitor ML352: Development of VU6001221, an improved in vivo tool compound.

Bertron JL, Ennis EA, Tarr CJ, Wright J, Dickerson JW, Locuson CW, Blobaum AL, Rook JM, Blakely RD, Lindsley CW
Bioorg Med Chem Lett. 2016 26 (19): 4637-4640

PMID: 27575469 · DOI:10.1016/j.bmcl.2016.08.062

MeSH Terms (11)

Animals Benzamides Dose-Response Relationship, Drug Half-Life Inhibitory Concentration 50 Isoxazoles Membrane Transport Proteins Oxazoles Piperidines Rats Structure-Activity Relationship

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