Discovery and characterization of a novel series of N-phenylsulfonyl-1H-pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu4).

Gogliotti RD, Blobaum AL, Morrison RM, Daniels JS, Salovich JM, Cheung YY, Rodriguez AL, Loch MT, Conn PJ, Lindsley CW, Niswender CM, Hopkins CR
Bioorg Med Chem Lett. 2016 26 (13): 2984-2987

PMID: 27234146 · PMCID: PMC4955388 · DOI:10.1016/j.bmcl.2016.05.029

MeSH Terms (10)

Allosteric Regulation Animals Microsomes, Liver Picolinic Acids Pyrroles Rats Receptors, Metabotropic Glutamate Structure-Activity Relationship Sulfonamides Triazoles

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