Novel GlyT1 inhibitor chemotypes by scaffold hopping. Part 2: development of a [3.3.0]-based series and other piperidine bioisosteres.

Sheffler DJ, Nedelcovych MT, Williams R, Turner SC, Duerk BB, Robbins MR, Jadhav SB, Niswender CM, Jones CK, Conn PJ, Daniels RN, Lindsley CW
Bioorg Med Chem Lett. 2014 24 (4): 1062-6

PMID: 24462664 · PMCID: PMC3951244 · DOI:10.1016/j.bmcl.2014.01.011

MeSH Terms (7)

Dose-Response Relationship, Drug Glycine Plasma Membrane Transport Proteins Humans Molecular Structure Piperidines Structure-Activity Relationship Sulfonamides

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