Synthesis and SAR of analogs of the M1 allosteric agonist TBPB. Part II: Amides, sulfonamides and ureas--the effect of capping the distal basic piperidine nitrogen.

Miller NR, Daniels RN, Bridges TM, Brady AE, Conn PJ, Lindsley CW
Bioorg Med Chem Lett. 2008 18 (20): 5443-7

PMID: 18829311 · PMCID: PMC3177607 · DOI:10.1016/j.bmcl.2008.09.032

MeSH Terms (15)

Allosteric Regulation Allosteric Site Amides Benzimidazoles Chemistry, Pharmaceutical Dose-Response Relationship, Drug Drug Design Humans Models, Chemical Nitrogen Piperidines Receptor, Muscarinic M1 Structure-Activity Relationship Sulfonamides Urea

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