Acyl dihydropyrazolo[1,5-a]pyrimidinones as metabotropic glutamate receptor 5 positive allosteric modulators.Malosh C, Turlington M, Bridges TM, Rook JM, Noetzel MJ, Vinson PN, Steckler T, Lavreysen H, Mackie C, Bartolomé-Nebreda JM, Conde-Ceide S, Martínez-Viturro CM, Piedrafita M, Sánchez-Casado MR, Macdonald GJ, Daniels JS, Jones CK, Niswender CM, Conn PJ, Lindsley CW, Stauffer SR
(2015)
Bioorg Med Chem Lett 25: 5115-20
MeSH Terms: Allosteric Regulation, Animals, Brain, Dogs, Humans, Ligands, Male, Motor Activity, Pyrazoles, Pyrimidines, Pyrimidinones, Rats, Rats, Sprague-Dawley, Receptor, Metabotropic Glutamate 5, Structure-Activity RelationshipAdded February 18, 2016